Methyldrostanolone, also known as methasteron, is a potent oral anabolic steroid that was never sold as a prescription drug. In structure, this steroid is a close derivative of drostanolone (Masteron). The only difference in this case is the addition of a c-17 alpha methyl group, a modification that gives this steroid high oral bioavailability.
The two agents remain very comparable, however. Both methyldrostanolone and drostanolone are non-aromatizable, so there is no difference in the estrogenicity of these two steroids, and both steroids retain favorable anabolic to androgenic ratios.
Methyldrostanolone is favored by athletes for its moderate anabolic properties, which are usually accompanied by fat loss and minimal androgenic side effects.
Brand name | Superdrol, Methyldrostonolone | |||
AndrogenicRatio | 20 | |||
AnabolicRatio | 400 | |||
Standard | Methyltestosterone (oral |
Superdrol Side Effects (Estrogenic)
Methyldrostanolone is not aromatized by the body, and is not measurably estrogenic. An anti-estrogen is not necessary when using this steroid, as gynecomastia should not be a concern even among sensitive individuals. Since estrogen is the usual culprit with water retention, methyldrostanolone instead produces a lean, quality look to the physique with no fear of excess subcutaneous fluid retention. This makes it a favorable steroid to use during cutting cycles, when water and fat retention are major concerns.
Superdrol Side Effects (Androgenic)
Although classified as an anabolic steroid, androgenic side effects are still possible with this substance, especially with higher doses. This may include bouts of oily skin, acne, and body/facial hair growth. Anabolic/androgenic steroids may also aggravate male pattern hair loss.
Women are warned of the potential virilizing effects of anabolic/androgenic steroids. These may include a deepening of the voice, menstrual irregularities, changes in skin texture, facial hair growth, and clitoral enlargement.
Superdrol Side Effects (Hepatotoxicity)
Methyldrostanolone is a c7-alpha alkylated compound. This alteration protects the drug from deactivation by the liver, allowing a very high percentage of the drug entry into the bloodstream following oral administration. Prolonged or high exposure may result in liver damage. In rare instances life-threatening dysfunction may develop. It is advisable to visit a physician periodically during each cycle to monitor liver function and overall health.
Note that although no human data can be found to make reference of, doses of 10 mg and 20 mg per day have been sufficient to produce high elevations of liver enzymes in consumers, as reported by private lab test results. Also, a small number of serious adverse events relating to liver toxicity have been reported with the use of this substance. The use of a liver detoxification supplement such as Lipid Stabil, Liv-52 is advised while taking any hepatotoxic anabolic/androgenic steroids.
Superdrol Side Effects (Cardiovascular)
To help reduce cardiovascular strain it is advised to maintain an active cardiovascular exercise program and minimize the intake of saturated fats, cholesterol, and simple carbohydrates at all times during active AAS administration. Supplementing with fish oils (4 grams per day) and a natural cholesterol/antioxidant formula such as Lipid Stabil .or a product with comparable ingredients is also recommended.
Superdrol Side Effects (Testosterone Suppression)
All anabolic/androgenic steroids when taken in doses sufficient to promote muscle gain are expected to suppress endogenous testosterone production. Without the intervention of testosterone-stimulating substances, testosterone levels should return to normal within 1-4 months of drug secession. Note that prolonged hypogonadotrophic hypogonadism can develop secondary to steroid abuse, necessitating medical intervention.
Superdrol Administration (Men)
Methydrostanolone was never approved for use in humans. Prescribing guidelines are unavailable. An effective dosage of methyldrostanolone for physique- or performance-enhancing purposes seems to begin in the range of 10-20 mg per day, taken for no longer than 6 or 8 weeks. At this level it seems to impart a measurable muscle-building effect, which is usually accompanied by fat loss and increased definition. Many do walk away with more than 10 pounds of solid muscle gain when using this agent alone.
In determining an optimal daily dosage, some do find the drug to be measurably more effective when venturing up to the 30 mg range. Potential hepatotoxicity should definitely be taken into account with such use, however. To avoid further escalating liver strain, 20 mg daily of methyldrostanolone is sometimes stacked with a nontoxic injectable steroid, such as testosterone for massbuilding phases of training, or nandrolone or boldenone for more lean tissue gain and definition, instead of simply increasing the dosage. The drug also works well in cutting cycles, where its lack of estrogenicity is highly favored. Often it is combined here with a non-aromatizable injectable steroid like Primobolan or Parabolan.
Superdrol Administration (Women)
Methyldrostanolone was never approved for use in humans. Prescribing guidelines are unavailable. In the athletic arena, an effective oral daily dosage would fall around 2.5 mg per day, taken in cycles lasting no more than 4-6 weeks to minimize the chance for virilization. The main point of contention with females is probably going to be the 10 mg per capsule dosage, which is far too high to use. Application would require opening each capsule and splitting the powdered contents up into 4 separate doses. As with all steroids, virilization is still possible.